SCHEMBL4253057

SCHEMBL4253057

N[C@@H]1CCC[C@@H]1c1cccc(F)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
GRIA4 P48058 1/20 0.49
TAAR1 Q96RJ0 1/20 0.44
KDM1A O60341 6/20 0.41
NOS3 P29474 2/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
RCOR1 Q9UKL0 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
P2RX7 Q99572 2/20 0.39
RIPK1 Q13546 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1645497 1.00 HTR2A (0.50) HTR2AHTR2CHTR2BGRIA4TAAR1
SCHEMBL1645763 0.96 HTR2A (0.50) HTR2AHTR2CHTR2BGRIA4TAAR1
SCHEMBL1645762 0.96 HTR2A (0.50) HTR2AHTR2CHTR2BGRIA4TAAR1
SCHEMBL3717272 0.81 GRIA4 (0.44) GRIA4KDM1ANOS3NOS1NOS2
SCHEMBL3717270 0.81 GRIA4 (0.44) GRIA4KDM1ANOS3NOS1NOS2
SCHEMBL1643845 0.81 GRIA4 (0.44) GRIA4KDM1ANOS3NOS1NOS2
SCHEMBL3719897 0.81 GRIA4 (0.44) GRIA4KDM1ANOS3NOS1NOS2
SCHEMBL3422301 0.81 HTR2C (0.61) HTR2AHTR2CHTR2BTAAR1KDM1A
SCHEMBL6998583 0.81 HTR2C (0.61) HTR2AHTR2CHTR2BTAAR1KDM1A
SCHEMBL3419759 0.81 HTR2C (0.61) HTR2AHTR2CHTR2BTAAR1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833782-B1 CYCLOALKYLAMINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-04-08 EP disclosed
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP disclosed