SCHEMBL4254835

SCHEMBL4254835

CN(C)c1ccc(N2Cc3ccc(F)cc3C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
PKM P14618 3/20 0.44
GAA P10253 2/20 0.42
UGCG Q16739 2/20 0.40
ADAM17 P78536 1/20 0.38
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
PGR P06401 1/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
DRD1 P21728 1/20 0.38
HTT P42858 1/20 0.38
NFKB2 Q00653 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4258064 0.89 PARP1 (0.46) PARP1NPC1RAB9APKMGAA
SCHEMBL4257849 0.84 NPC1 (0.56) PARP1NPC1RAB9APKMGAA
SCHEMBL4250602 0.83 HTR2C (0.47) PARP1NPC1RAB9APKMGAA
SCHEMBL4258304 0.80 NPC1 (0.69) PARP1NPC1RAB9APKMGAA
SCHEMBL4253350 0.79 NPC1 (0.48) NPC1RAB9APKMGAAUGCG
SCHEMBL1468586 0.78 NPC1 (0.47) PARP1NPC1RAB9APKMGAA
SCHEMBL1468585 0.76 NPC1 (0.41) PARP1NPC1RAB9APKMGAA
SCHEMBL4250783 0.76 NPC1 (0.56) PARP1NPC1RAB9APKMGAA
SCHEMBL10085886 0.76 NPC1 (0.70) NPC1RAB9APKMGAATP53
SCHEMBL4255757 0.75 PARP1 (0.49) PARP1NPC1RAB9APKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed