SCHEMBL4257312

SCHEMBL4257312

O=C(Nc1cc(-c2ccccc2)ccc1[AsH2])c1ccc(N2CCC3(CCN(c4ccccc4)C3)C2)nc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 19/20 0.59
HDAC1 Q13547 18/20 0.59
HDAC2 Q92769 4/20 0.59
HDAC3 O15379 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1640709 0.90 HDAC1 (0.73) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1639127 0.82 HDAC1 (0.75) KCNH2HDAC1HDAC2HDAC3
SCHEMBL3621838 0.81 HDAC1 (0.71) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1639782 0.81 HDAC1 (0.73) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1640955 0.80 HDAC1 (0.79) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1639868 0.80 HDAC1 (0.69) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1640882 0.79 HDAC1 (0.69) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1639698 0.79 HDAC1 (0.67) KCNH2HDAC1HDAC2HDAC3
SCHEMBL13811465 0.78 HDAC1 (0.90) KCNH2HDAC1HDAC2HDAC3
SCHEMBL1640470 0.78 HDAC1 (0.82) KCNH2HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954698-B1 SPIROCYCLIC COMPOUNDS AS HDAC INHIBITORS MERCK & CO INC (US) 2009-06-24 EP disclosed