SCHEMBL4257489

SCHEMBL4257489

CC(C)(C)/C(=C\C(=O)O)c1ccc(C(=C2CCCCCC2)c2cccc(O)c2)cc1F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA6 P23280 1/20 0.33
CA9 Q16790 1/20 0.33
ESR1 P03372 4/20 0.33
RXRA P19793 2/20 0.33
RXRB P28702 2/20 0.33
RXRG P48443 2/20 0.33
HSD17B1 P14061 2/20 0.33
HSD17B2 P37059 2/20 0.33
SLC2A1 P11166 1/20 0.33
SLC2A4 P14672 1/20 0.33
PGR P06401 1/20 0.33
CHRM2 P08172 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
AR P10275 1/20 0.33
CHRM1 P11229 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256094 0.90 ESR1 (0.40) ESR1RXRARXRBRXRGPGR
SCHEMBL4262517 0.87 ESR1 (0.39) CA12CA1CA2CA6CA9
SCHEMBL4258861 0.82 ESR1 (0.38) ESR1RXRARXRBRXRGPGR
SCHEMBL4253218 0.80 ESR1 (0.42) ESR1RXRARXRBPGRCHRM2
SCHEMBL4254771 0.79 ESR1 (0.39) ESR1RXRAPGRCHRM2ADORA3
SCHEMBL4257498 0.78 CA12 (0.33) CA12CA1CA2CA6CA9
SCHEMBL3468460 0.76 MIF (0.54) CA12CA1CA2CA6CA9
SCHEMBL3468457 0.76 MIF (0.54) CA12CA1CA2CA6CA9
SCHEMBL4257434 0.75 ESR1 (0.47) CA12CA1CA2CA6CA9
SCHEMBL4258950 0.75 ESR1 (0.47) CA12CA1CA2CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7569601-B2 Cycloalkylidene compounds as modulators of estrogen receptor SMITHKLINE BEECHAM CORPORATION (US) 2009-08-04 US disclosed
US-20070213348-A1 Chemical Compounds BRITTON JONATHAN E 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213348-A1 Chemical Compounds GPER1, ESR2, ESR1 CA12 2173/4885CA1 2385/4885CA2 1998/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.