SCHEMBL4258682

SCHEMBL4258682

CC(Nc1ncc(C#N)c(-c2cnc3c(Cl)cccn23)n1)c1ccc([C@@H](O)CNC(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 4/20 0.35
PLK1 P53350 4/20 0.35
ADRB2 P07550 2/20 0.33
ADRB1 P08588 2/20 0.33
CYP2D6 P10635 1/20 0.33
NFKB1 P19838 1/20 0.33
HIF1A Q16665 1/20 0.33
BLM P54132 1/20 0.32
HTR1A P08908 2/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
MAOA P21397 1/20 0.31
HTR2B P41595 1/20 0.31
CDK1 P06493 1/20 0.31
KDR P35968 1/20 0.31
MAP3K8 P41279 2/20 0.31
CDK2 P24941 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3R2 O00459 1/20 0.31
PIK3CG P48736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200557 1.00 IGF1R (0.35) IGF1RPLK1ADRB2ADRB1CYP2D6
SCHEMBL2198357 1.00 IGF1R (0.35) IGF1RPLK1ADRB2ADRB1CYP2D6
SCHEMBL2197154 1.00 IGF1R (0.35) IGF1RPLK1ADRB2ADRB1CYP2D6
SCHEMBL2198544 0.91 PLK1 (0.35) IGF1RPLK1HTR1AADRA2AADRA2B
SCHEMBL2198979 0.90 IGF1R (0.38) IGF1RADRB2ADRB1CYP2D6NFKB1
SCHEMBL2196563 0.90 PLK1 (0.34) IGF1RPLK1HTR1AADRA2AADRA2B
SCHEMBL19951497 0.90 PLK1 (0.34) IGF1RPLK1HTR1AADRA2AADRA2B
SCHEMBL4272407 0.90 PLK1 (0.34) IGF1RPLK1HTR1AADRA2AADRA2B
SCHEMBL4264314 0.90 PLK1 (0.34) IGF1RPLK1HTR1AADRA2AADRA2B
SCHEMBL2198389 0.90 PLK1 (0.34) IGF1RPLK1HTR1AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2116543-A1 NOVEL AMINOPYRIMIDINE DERIVATIVE AS PLK1 INHIBITOR BANYU PHARMACEUTICAL CO., LTD. (JP) 2009-11-11 EP disclosed