SCHEMBL4274589

SCHEMBL4274589

Cc1c(Sc2ccc(S(C)(=O)=O)cc2)c2cc(-c3ccsc3)ccc2n1CC(=O)O.Cc1c(Sc2ccc(S(C)(=O)=O)cc2)c2cc(-c3cncnc3)ccc2n1CC(=O)O

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.63
AKR1B1 P15121 9/20 0.63
CYP2C9 P11712 3/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1252422 0.93 PTGDR2 (0.72) PTGDR2AKR1B1CYP2C9
SCHEMBL2549980 0.93 PTGDR2 (0.72) PTGDR2AKR1B1CYP2C9
SCHEMBL1251040 0.92 PTGDR2 (0.54) PTGDR2AKR1B1CYP2C9
SCHEMBL1251019 0.84 PTGDR2 (0.68) PTGDR2AKR1B1CYP2C9
SCHEMBL5731063 0.82 PTGDR2 (0.43) PTGDR2AKR1B1CYP2C9
SCHEMBL4274593 0.82 PTGDR2 (0.56) PTGDR2AKR1B1CYP2C9
SCHEMBL1251026 0.80 PTGDR2 (0.68) PTGDR2AKR1B1CYP2C9
SCHEMBL12913905 0.80 PTGDR2 (0.59) PTGDR2AKR1B1CYP2C9
SCHEMBL5732122 0.80 PTGDR2 (0.54) PTGDR2AKR1B1CYP2C9
SCHEMBL1252380 0.79 PTGDR2 (0.69) PTGDR2AKR1B1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2025670-A1 3-(Phenyl or quinolyl)thio-1H-indole-1-acetic acid derivatives as modulators of CRTh2 receptor activity AstraZeneca AB (SE) 2009-02-18 EP disclosed