SCHEMBL4277571

SCHEMBL4277571

[CH2]c1nc2c(oc3ccc(Br)cc32)c(=O)[nH]1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CSNK2B P67870 20/20 0.64
PIM1 P11309 19/20 0.64
CDC7 O00311 9/20 0.64
CSNK2A1 P68400 9/20 0.64
CSNK2A2 P19784 13/20 0.60
PIM3 Q86V86 12/20 0.60
PIM2 Q9P1W9 12/20 0.60
CSNK2A3 Q8NEV1 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12661564 0.83 CSNK2B (0.67) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1856877 0.83 CSNK2B (0.67) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1853268 0.81 CSNK2B (0.67) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1854454 0.80 CSNK2B (0.69) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1857243 0.80 CSNK2B (0.63) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1850855 0.80 PIM1 (0.69) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1852949 0.79 CSNK2B (0.58) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1853281 0.78 CSNK2B (1.00) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1854480 0.78 CSNK2B (1.00) CSNK2BPIM1CDC7CSNK2A1CSNK2A2
SCHEMBL1849054 0.78 CSNK2B (1.00) CSNK2BPIM1CDC7CSNK2A1CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097419-A1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS Exelixis, Inc. (US) 2009-09-09 EP disclosed
WO-2009086264-A1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS EXELIXIS, INC. (US) 2009-07-09 WO disclosed