SCHEMBL4281796

SCHEMBL4281796

O=CCc1cccc(-c2cc(Nc3ccc(OC(F)(F)F)cc3)cc(N3CCOCC3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 6/20 0.48
BCR P11274 5/20 0.48
CTSS P25774 3/20 0.44
CTSK P43235 2/20 0.44
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
MCHR1 Q99705 1/20 0.43
KCNH2 Q12809 1/20 0.43
AKT1 P31749 2/20 0.42
PIK3CA P42336 3/20 0.42
MTOR P42345 1/20 0.41
PIM1 P11309 1/20 0.41
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5183368 0.86 PIK3CA (0.58) ABL1BCRCTSSCTSKPIK3CA
SCHEMBL5182531 0.85 ABL1 (0.55) ABL1BCRCTSSCTSKRAF1
SCHEMBL4358479 0.83 ABL1 (0.55) ABL1BCRCTSSCTSKRAF1
SCHEMBL3996650 0.83 ABL1 (0.56) ABL1BCRCTSSCTSKRAF1
SCHEMBL3997711 0.81 ABL1 (0.63) ABL1BCRRAF1BRAFMCHR1
SCHEMBL4361850 0.81 NPSR1 (0.53) AKT1PIK3CAMTORCYP1A2CYP3A4
SCHEMBL4358342 0.81 ABL1 (0.56) ABL1BCRCTSSCTSKMCHR1
SCHEMBL4004651 0.75 ABL1 (0.61) ABL1BCRCTSSCTSKRAF1
SCHEMBL4358482 0.75 ABL1 (0.58) ABL1BCRRAF1BRAFMCHR1
SCHEMBL3450413 0.75 ABL1 (0.56) ABL1BCRCTSSCTSKRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805142-A4 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS INC (US) 2009-06-10 EP disclosed
EP-1805142-A2 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM Reddy US Therapeutics, Inc. (US) 2007-07-11 EP disclosed
WO-2006034474-A2 NOVEL PYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS, INC. (US) 2006-03-30 WO disclosed