SCHEMBL4286092

SCHEMBL4286092

NC(=O)Oc1ccc(-c2nc3c(oc4ccc(Br)cc43)c(=O)[nH]2)c(Cl)c1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 19/20 0.71
CSNK2A2 P19784 19/20 0.71
CSNK2B P67870 19/20 0.71
PIM3 Q86V86 18/20 0.71
PIM2 Q9P1W9 18/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1850345 0.87 CSNK2A2 (0.76) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1855496 0.86 PIM1 (0.89) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1852355 0.83 PIM1 (0.80) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1854063 0.83 PIM1 (1.00) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1852633 0.81 CSNK2A2 (0.71) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1849631 0.81 PIM1 (1.00) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1851595 0.81 PIM1 (1.00) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1852531 0.80 PIM1 (0.72) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL13650454 0.80 PIM1 (0.68) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1850401 0.80 CSNK2A2 (1.00) PIM1CSNK2A2CSNK2BPIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097419-A1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS Exelixis, Inc. (US) 2009-09-09 EP disclosed
WO-2009086264-A1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS EXELIXIS, INC. (US) 2009-07-09 WO disclosed