SCHEMBL4288458

SCHEMBL4288458

COc1ccc(C)c(-c2cc(Cl)nc(N)n2)c1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.76
HSP90AB1 P08238 11/20 0.76
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
AGPAT2 O15120 3/20 0.47
NPC1 O15118 2/20 0.46
ADCY10 Q96PN6 1/20 0.46
DYRK1A Q13627 1/20 0.44
KDM4E B2RXH2 1/20 0.44
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3946976 0.87 HSP90AA1 (1.00) HSP90AA1HSP90AB1POLBGAAMAPT
SCHEMBL3942089 0.85 HSP90AA1 (0.76) HSP90AA1HSP90AB1POLBGAAMAPT
SCHEMBL3945098 0.84 HSP90AA1 (1.00) HSP90AA1HSP90AB1POLBGAAMAPT
SCHEMBL4282884 0.81 AGPAT2 (0.67) HSP90AA1HSP90AB1AGPAT2KDM4E
SCHEMBL4282163 0.81 HSP90AA1 (0.54) HSP90AA1HSP90AB1AGPAT2DYRK1AKDM4E
SCHEMBL2849242 0.81 HSP90AA1 (0.52) HSP90AA1HSP90AB1AGPAT2KDM4E
SCHEMBL2850401 0.79 BACE1 (0.52) HSP90AA1HSP90AB1GAAMAPTSMN1; SMN2
SCHEMBL13880245 0.79 AGPAT2 (0.79) POLBGAAMAPTSMN1; SMN2AGPAT2
SCHEMBL4289224 0.79 AGPAT2 (0.64) HSP90AA1HSP90AB1MAPTAGPAT2ADCY10
SCHEMBL2849100 0.79 AGPAT2 (0.64) HSP90AA1HSP90AB1AGPAT2NPC1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090099183-A1 PYRIMIDINES AND USES THEREOF CELL THERAPEUTICS, INC. (US) 2009-04-16 US disclosed
US-7419984-B2 Pyrimidines and uses thereof CELL THERAPEUTICS, INC. (US) 2008-09-02 US disclosed
US-20040204386-A1 Pyrimidines and uses thereof CELL THERAPEUTICS, INC. 2004-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040204386-A1 Pyrimidines and uses thereof LPCAT3, LPCAT1, APRT HSP90AA1 4126/4885HSP90AB1 4236/4885POLB 443/4885
US-20090099183-A1 PYRIMIDINES AND USES THEREOF LPCAT3, LPCAT1, APRT HSP90AA1 4006/4885HSP90AB1 3829/4885POLB 257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.