SCHEMBL4295879

SCHEMBL4295879

CC(C)S(=O)(=O)NC[C@@](C)(F)c1ccc(I)cc1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 12/20 0.46
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
GRIA1 P42261 3/20 0.33
TRPV1 Q8NER1 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4295881 1.00 GRIA4 (0.46) GRIA4CA1CA2GRIA1TRPV1
SCHEMBL6561639 0.92 GRIA4 (0.51) GRIA4CA1CA2GRIA1CA12
SCHEMBL3711628 0.88 GRIA4 (0.48) GRIA4CA1CA2GRIA1
SCHEMBL13255710 0.88 GRIA4 (0.48) GRIA4CA1CA2GRIA1
SCHEMBL5186065 0.82 GRIA4 (0.43) GRIA4CA1CA2
SCHEMBL5186189 0.82 GRIA4 (0.54) GRIA4GRIA1
SCHEMBL5769048 0.82 GRIA4 (0.42) GRIA4CA1CA2GRIA1CA12
SCHEMBL3703932 0.82 CYP2C19 (0.47) GRIA4CA1CA2GRIA1
SCHEMBL3703930 0.82 CYP2C19 (0.47) GRIA4CA1CA2GRIA1
SCHEMBL13663202 0.81 GRIA4 (0.43) GRIA4CA1CA2GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010087982-A1 GLUR2 RECEPTOR MODULATORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2010-08-05 WO disclosed
US-20090270508-A1 GluR2 receptor modulators NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2009-10-29 US disclosed
US-20090270508-A1 GluR2 receptor modulators NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2009-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270508-A1 GluR2 receptor modulators GRM2, GRIK2, GRIN2A GRIA4 16/4885CA1 1934/4885CA2 1890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.