SCHEMBL4299699

SCHEMBL4299699

O=C(O)C1=CN(C(=O)c2ccc(F)cc2)C(C(=O)O)Cc2c1[nH]c1ccccc21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.48
ABCB1 P08183 2/20 0.45
ABCG2 Q9UNQ0 2/20 0.45
CDK4 P11802 1/20 0.44
CCND1 P24385 1/20 0.44
CYP19A1 P11511 2/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
ACE P12821 1/20 0.40
DRD5 P21918 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4300714 0.92 CYP19A1 (0.45) ABCB1ABCG2CYP19A1ALDH1A1TSHR
SCHEMBL687916 0.87 NR1H4 (0.50) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL29880554 0.87 NR1H4 (0.50) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL328164 0.86 NR1H4 (0.49) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL4300281 0.82 HSD17B10 (0.47) ALDH1A1TSHR
SCHEMBL4302795 0.79 ABCG2 (0.43) NR1H4ABCB1ABCG2
SCHEMBL274449 0.79 NR1H4 (0.67) NR1H4ALDH1A1
SCHEMBL273514 0.79 NR1H4 (0.67) NR1H4ALDH1A1
SCHEMBL275134 0.79 NR1H4 (0.67) NR1H4ALDH1A1
SCHEMBL5733404 0.78 NR1H4 (0.49) NR1H4ABCB1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7595311-B2 Modulating active of receptors; therapy prevention of disease such aas symthrome X, antidiabetic agents, insulin resistance, hypoglycemic agents EXELIXIS, INC. (US) 2009-09-29 US claimed
CN-110404073-B Methods and pharmaceutical compositions for treating hepatitis B virus infection 国家医疗保健研究所 2022-08-16 CN disclosed