SCHEMBL4300282

SCHEMBL4300282

Cc1nc(Cl)cc2c(Cl)c(C(N)=O)cnc12

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.54
PARP1 P09874 7/20 0.41
NNMT P40261 5/20 0.40
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
PIM1 P11309 1/20 0.38
TTK P33981 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
BTK Q06187 1/20 0.35
POLB P06746 1/20 0.34
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321604 0.75 SLC2A1 (0.63) SLC2A1PARP1NNMTRXFP1PIM1
SCHEMBL4625947 0.74 SLC2A1 (0.77) SLC2A1PARP1NNMTPIM1TTK
SCHEMBL7622343 0.74 SLC2A1 (0.50) SLC2A1PARP1NNMTPIM1TTK
SCHEMBL2483995 0.72 NPSR1 (0.50) SLC2A1PARP1NNMTNPSR1RXFP1
SCHEMBL5464747 0.70 SLC2A1 (0.56) SLC2A1NNMTRXFP1MEN1KMT2A
SCHEMBL15054260 0.70 SLC2A1 (0.47) SLC2A1PARP1NNMTNPSR1RXFP1
SCHEMBL17646064 0.70 SLC2A1 (0.50) SLC2A1PARP1NNMTNPSR1RXFP1
SCHEMBL3965438 0.70 SLC2A1 (0.47) SLC2A1PARP1NNMTPDE4B
SCHEMBL31251385 0.70 KMT2A (0.59) MEN1KMT2APOLB
SCHEMBL12876619 0.69 SLC2A1 (0.46) SLC2A1NNMTPIM1TTKPIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090270444-A1 1,7-Naphthyridines GLAXO GROUP LIMITED (GB) 2009-10-29 US disclosed
US-20090270444-A1 1,7-Naphthyridines GLAXO GROUP LIMITED (GB) 2009-10-29 US disclosed
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors GLAXO GROUP LIMITED 2008-06-19 US disclosed
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors GLAXO GROUP LIMITED 2008-06-19 US disclosed
EP-1866305-A1 1,7-NAPHTHYRIDINES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2007-12-19 EP disclosed
EP-1812434-A2 1,7-NAPHTHYRIDINES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2007-08-01 EP disclosed
WO-2006097340-A1 1,7-NAPHTHYRIDINES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2006-09-21 WO disclosed
WO-2006097340-A1 1,7-NAPHTHYRIDINES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2006-09-21 WO disclosed
WO-2006053784-A2 1,7-NAPHTHYRIDINES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2006-05-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors PDE4A, PDE3B, PDE4B SLC2A1 3875/4885PARP1 1580/4885NNMT 83/4885
US-20090270444-A1 1,7-Naphthyridines CYP2F1, CYP2S1, CYP1A1 SLC2A1 1779/4885PARP1 1391/4885NNMT 2350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.