SCHEMBL4303476

SCHEMBL4303476

O=C1CN(c2ccc(-c3ccsc3)cc2O)S(=O)(=O)N1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 10/20 0.61
ERN1 O75460 2/20 0.40
ACMSD Q8TDX5 1/20 0.40
PTPN2 P17706 6/20 0.38
PTPRC P08575 1/20 0.35
CHEK1 O14757 1/20 0.34
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12056201 0.88 PTPN1 (0.74) PTPN1PTPN2
SCHEMBL3918247 0.82 PTPN1 (0.70) PTPN1ACMSDPTPN2ALOX5
SCHEMBL3221334 0.80 PTPN1 (0.57) PTPN1PTPN2CHEK1
SCHEMBL3920603 0.80 PTPN1 (0.67) PTPN1PTPN2
SCHEMBL3222925 0.79 PTPN1 (0.65) PTPN1PTPN2
SCHEMBL3918842 0.78 PTPN1 (0.61) PTPN1ERN1PTPN2CHEK1
SCHEMBL3214144 0.77 PTPN1 (0.60) PTPN1PTPN2CHEK1
SCHEMBL3926871 0.76 PTPN1 (0.58) PTPN1PTPN2
SCHEMBL3224416 0.76 PTPN1 (0.58) PTPN1PTPN2
SCHEMBL3928767 0.76 ERN1 (0.40) PTPN1ERN1ACMSDPTPRCCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
WO-2007115058-A2 THIADIAZOLIDINONE INHIBITORS OF PTPASE NOVARTIS AG (CH) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181928-A1 ORGANIC COMPOUNDS PTPRS, PTPRO, PTPRC PTPN1 21/4885ERN1 3193/4885ACMSD 4777/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.