SCHEMBL4318238

SCHEMBL4318238

Cc1c(-c2ccc(F)c(C(F)(F)F)c2)n(CC(=O)NC(C)(C)C)c(=O)c2cc(O)cn12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 2/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 2/20 0.38
NPC1 O15118 1/20 0.38
GRIN2B Q13224 7/20 0.37
GRIN1 Q05586 3/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
TRPA1 O75762 1/20 0.36
NR1I2 O75469 1/20 0.35
CSNK1D P48730 1/20 0.35
CSNK1E P49674 1/20 0.35
CNR2 P34972 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4302713 0.89 AVPR1B (0.44) AVPR1BLMNAGAANPC1GRIN2B
SCHEMBL4309843 0.88 AVPR1B (0.52) AVPR1BGRIN2BGRIN1ALDH1A1KDM4E
SCHEMBL4304952 0.82 AVPR1B (0.63) AVPR1B
SCHEMBL8013549 0.77 AVPR1B (0.56) AVPR1BGRIN2B
SCHEMBL4308725 0.72 AVPR1B (0.75) AVPR1B
SCHEMBL4309710 0.70 AVPR1B (0.50) AVPR1B
SCHEMBL4311095 0.70 AVPR1B (0.68) AVPR1B
SCHEMBL4301376 0.70 AVPR1B (0.66) AVPR1BLMNAGRIN2BGRIN1NR1I2
SCHEMBL4315024 0.66 AVPR1B (0.84) AVPR1B
SCHEMBL4306581 0.62 AVPR1B (0.67) AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed