SCHEMBL4332779

SCHEMBL4332779

CC(NC(=O)C1c2ccccc2C(=O)N1C1CNC1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.58
SCN5A Q14524 13/20 0.58
KCNH2 Q12809 13/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13577793 0.88 SCN9A (0.70) SCN9ASCN5AKCNH2
SCHEMBL13577794 0.85 SCN9A (0.73) SCN9ASCN5AKCNH2
SCHEMBL4321096 0.82 SCN9A (0.80) SCN9ASCN5AKCNH2
Trifluoroacetic Acid SCHEMBL4337866 0.79 SCN9A (0.75) SCN9ASCN5AKCNH2
SCHEMBL4476223 0.77 SCN9A (0.71) SCN9ASCN5AKCNH2
SCHEMBL4325532 0.74 SCN9A (0.80) SCN9ASCN5AKCNH2
SCHEMBL3892332 0.74 SCN9A (0.84) SCN9ASCN5AKCNH2
SCHEMBL4332708 0.73 SCN9A (1.00) SCN9ASCN5AKCNH2
SCHEMBL4323513 0.72 SCN9A (0.81) SCN9ASCN5AKCNH2
SCHEMBL4325285 0.72 SCN9A (1.00) SCN9ASCN5AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145721-A1 ISOINDOLINE DERIVATIVES COMPRISING PHENYL GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO claimed
WO-2009145721-A1 ISOINDOLINE DERIVATIVES COMPRISING PHENYL GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed