SCHEMBL4337689

SCHEMBL4337689

Cn1cc(-c2c(Cl)n(CCCC(=O)O)c3c(=O)[nH]cnc23)cn1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 1/20 0.38
PDK2 Q15119 4/20 0.35
BRD4 O60885 2/20 0.35
HPRT1 P00492 1/20 0.32
PNP P00491 1/20 0.32
AURKA O14965 1/20 0.32
TTK P33981 1/20 0.32
AURKB Q96GD4 1/20 0.32
INCENP Q9NQS7 1/20 0.32
EGLN1 Q9GZT9 2/20 0.32
HSD17B10 Q99714 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PDPK1 O15530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4325427 0.85 ACVR1 (0.36) ACVR1PDK2BRD4HPRT1PNP
SCHEMBL4337687 0.83 KDM4E (0.44) BRD4HSD17B10KDM4EPOLB
SCHEMBL4339090 0.67 BACE1 (0.42) EGLN1ALDH1A1
SCHEMBL4337751 0.63 BRD4 (0.41) PDK2BRD4HSD17B10
SCHEMBL22084778 0.62 SRC (0.48) ACVR1BRD4AURKAAURKBINCENP
SCHEMBL15845784 0.62 ACVR1 (0.63) ACVR1BRD4AURKATTKAURKB
SCHEMBL4213891 0.61 HRH3 (0.49) HSD17B10
SCHEMBL16663845 0.60 ACVR1 (0.42) ACVR1PDK2BRD4AURKATTK
SCHEMBL32689791 0.58 PLAU (0.47) AURKAAURKBEGLN1ALDH1A1
SCHEMBL8237863 0.58 HPGD (0.38) BRD4HSD17B10KDM4EALDH1A1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7557113-B2 Substituted pyrrolo[3,2-d]pyrimidine derivatives TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
US-7557113-B2 Substituted pyrrolo[3,2-d]pyrimidine derivatives TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
US-7557113-B2 Substituted pyrrolo[3,2-d]pyrimidine derivatives TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
EP-1661897-A1 PYRROLOPYRIMIDINONE DERIVATIVE Teijin Pharma Limited (JP) 2006-05-31 EP disclosed