SCHEMBL4339344

SCHEMBL4339344

CCCc1onc(COc2c(C)cccc2C)c1COc1ccc(-c2ccc3nc(C(=O)OC)ccc3c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 19/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4336901 0.92 NR1H4 (0.53) NR1H4CYP1A2CYP2C9
SCHEMBL4332220 0.90 NR1H4 (0.46) NR1H4CYP1A2CYP2C9MEN1KMT2A
SCHEMBL4335327 0.89 NR1H4 (0.46) NR1H4CYP1A2CYP2C9
SCHEMBL2000357 0.87 NR1H4 (0.57) NR1H4CYP1A2CYP2C9
SCHEMBL4341584 0.84 NR1H4 (0.53) NR1H4CYP1A2CYP2C9
SCHEMBL4330187 0.84 NR1H4 (0.42) NR1H4CYP1A2CYP2C9
SCHEMBL4332197 0.83 NR1H4 (0.60) NR1H4CYP1A2CYP2C9
SCHEMBL4337574 0.82 NR1H4 (0.65) NR1H4CYP1A2CYP2C9
SCHEMBL4339455 0.81 NR1H4 (0.48) NR1H4CYP1A2CYP2C9
SCHEMBL4332090 0.80 NR1H4 (0.49) NR1H4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079307-A2 FARNESOID X RECEPTOR AGONISTS SmithKline Beecham Corporation (US) 2009-07-22 EP disclosed
WO-2008051942-A2 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-05-02 WO disclosed