SCHEMBL4345514

SCHEMBL4345514

O=C(NCc1ccc(C(F)(F)F)cc1)N(S)c1cc(Cl)cc(CCO)c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.38
HDAC1 Q13547 2/20 0.38
LSS P48449 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPT P10636 1/20 0.37
MAPK14 Q16539 1/20 0.36
MEN1 O00255 1/20 0.36
PLA2G1B P04054 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4351483 0.86 MTOR (0.42) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4347804 0.81 KCNH2 (0.39) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4359745 0.81 TMPRSS4 (0.50) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4355927 0.77 LSS (0.44) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4347497 0.76 MAPT (0.47) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4357500 0.76 HDAC3 (0.46) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4345512 0.76 KMT2A (0.49) MAPTMEN1GAAKMT2AALDH1A1
SCHEMBL4354458 0.75 MTOR (0.42) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4354240 0.75 MTOR (0.43) MTORHDAC1LSSHDAC3HDAC2
SCHEMBL4348897 0.74 MTOR (0.50) MTORHDAC1LSSHDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed