SCHEMBL4350322

SCHEMBL4350322

CC(C)(C)CC(C)(C)NC(=O)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.50
HTT P42858 4/20 0.50
MAPT P10636 4/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
AR P10275 1/20 0.38
GAA P10253 3/20 0.38
TP53 P04637 2/20 0.38
EPHX1 P07099 2/20 0.38
THRB P10828 2/20 0.38
RECQL P46063 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PLEC Q15149 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344564 0.84 HTT (0.53) POLBHTTMAPTMEN1KMT2A
SCHEMBL4351163 0.82 HTT (0.58) POLBHTTMAPTMEN1KMT2A
SCHEMBL4341979 0.82 POLB (0.54) POLBHTTMAPTMEN1KMT2A
SCHEMBL4351212 0.82 POLB (0.56) POLBHTTMAPTMEN1KMT2A
SCHEMBL4346754 0.82 POLB (0.50) POLBHTTMAPTMEN1KMT2A
SCHEMBL4341316 0.81 MAPT (0.41) POLBHTTMAPTMEN1KMT2A
SCHEMBL4343991 0.79 HTT (0.40) POLBHTTMAPTMEN1KMT2A
SCHEMBL6568509 0.77 POLB (0.52) POLBHTTMAPTMEN1KMT2A
SCHEMBL4344549 0.76 POLB (0.48) POLBHTTMAPTMEN1KMT2A
SCHEMBL4342367 0.75 HTT (0.47) POLBHTTMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed