SCHEMBL4353358

SCHEMBL4353358

CC(C)(C)NC(=S)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 5/20 0.47
MEN1 O00255 3/20 0.47
GAA P10253 3/20 0.47
KMT2A Q03164 3/20 0.47
MAPT P10636 3/20 0.47
ALOX12 P18054 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 4/20 0.41
NPSR1 Q6W5P4 3/20 0.40
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
TNF P01375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4351212 0.82 POLB (0.56) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL9355759 0.81 HTT (0.53) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4347722 0.81 HTT (0.54) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4351163 0.79 HTT (0.58) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4343493 0.79 HTT (0.59) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4343700 0.79 HTT (0.50) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4358256 0.76 HTT (0.47) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL12404443 0.75 SMN1; SMN2 (0.71) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL4351130 0.75 KDM4E (0.45) HTTALDH1A1MEN1GAAKMT2A
SCHEMBL9355733 0.75 MAOB (0.53) HTTSMN1; SMN2ALDH1A1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed