SCHEMBL4354543

SCHEMBL4354543

CC(C)NC(=S)Nc1cc(Cl)c(O)c(-c2nc3ccccc3s2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.50
MAPT P10636 11/20 0.48
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 3/20 0.48
GAA P10253 2/20 0.48
MEN1 O00255 6/20 0.47
KMT2A Q03164 6/20 0.47
RAB9A P51151 4/20 0.47
THRB P10828 2/20 0.44
TP53 P04637 3/20 0.43
RXFP1 Q9HBX9 2/20 0.43
POLB P06746 2/20 0.43
NPC1 O15118 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
CTSD P07339 1/20 0.43
EGFR P00533 1/20 0.42
INSR P06213 1/20 0.42
IGF1R P08069 1/20 0.42
PDGFRB P09619 1/20 0.42
SRC P12931 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846512 0.89 SMN1; SMN2 (0.50) SMN1; SMN2MAPTALDH1A1KDM4EGAA
SCHEMBL4341725 0.85 MAPT (0.52) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL4502451 0.84 MAPT (0.50) SMN1; SMN2MAPTALDH1A1KDM4EGAA
SCHEMBL4348872 0.82 MEN1 (0.48) SMN1; SMN2MAPTALDH1A1KDM4EGAA
SCHEMBL4561504 0.80 MAPT (0.54) SMN1; SMN2MAPTALDH1A1KDM4EGAA
SCHEMBL4354538 0.80 SMN1; SMN2 (0.52) SMN1; SMN2MAPTKDM4EGAAMEN1
SCHEMBL4352804 0.78 MAPT (0.56) SMN1; SMN2MAPTALDH1A1KDM4EGAA
SCHEMBL6224490 0.77 MAPT (0.44) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL12846511 0.77 SMN1; SMN2 (0.49) SMN1; SMN2MAPTKDM4EMEN1KMT2A
SCHEMBL4341723 0.76 MAPT (0.49) SMN1; SMN2MAPTKDM4EGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed