SCHEMBL4354564

SCHEMBL4354564

O=C(Nc1cc(Cl)cc(Cl)c1)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
MAPT P10636 4/20 0.58
RAB9A P51151 3/20 0.58
NPSR1 Q6W5P4 1/20 0.58
P2RY1 P47900 1/20 0.54
LMNA P02545 4/20 0.49
ALDH1A1 P00352 2/20 0.49
SLC2A1 P11166 1/20 0.49
DHODH Q02127 1/20 0.47
HTT P42858 2/20 0.47
TRPV1 Q8NER1 1/20 0.46
S1PR2 O95136 1/20 0.46
NPC1 O15118 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
P2RX1 P51575 1/20 0.44
P2RX4 Q99571 1/20 0.44
P2RX7 Q99572 1/20 0.44
TMPRSS4 Q9NRS4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348841 0.86 MEN1 (0.57) MEN1KMT2AMAPTRAB9ALMNA
SCHEMBL15786287 0.84 MEN1 (0.76) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL4350046 0.84 MEN1 (0.49) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL4347321 0.83 P2RY1 (0.61) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL4348031 0.81 MAOB (0.64) MEN1KMT2AMAPTNPSR1LMNA
SCHEMBL4342271 0.81 KMT2A (0.53) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL29555610 0.81 MEN1 (0.61) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL4353624 0.81 P2RY1 (0.68) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL29556187 0.81 MEN1 (0.61) MEN1KMT2AMAPTRAB9ANPSR1
SCHEMBL4345397 0.79 TRPV1 (0.58) MEN1KMT2AMAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed