SCHEMBL4355870

SCHEMBL4355870

CC(C)(C)CC(C)(C)NC(=S)Nc1cc(Br)c(O)c(Br)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.56
POLB P06746 4/20 0.56
MAPT P10636 6/20 0.43
ALDH1A1 P00352 6/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
GAA P10253 3/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.42
NPSR1 Q6W5P4 2/20 0.40
GLA P06280 1/20 0.40
TNF P01375 1/20 0.40
NOD2 Q9HC29 1/20 0.40
NOD1 Q9Y239 1/20 0.40
ALOX12 P18054 3/20 0.37
HPGD P15428 3/20 0.37
CYP3A4 P08684 2/20 0.37
TSHR P16473 2/20 0.37
HIF1A Q16665 2/20 0.37
HSD17B10 Q99714 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4343493 0.82 HTT (0.59) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4345688 0.82 HTT (0.56) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4346754 0.82 POLB (0.50) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4351212 0.82 POLB (0.56) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL6669894 0.74 HTT (0.49) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4350392 0.73 HTT (0.44) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4343912 0.73 HTT (0.47) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4351871 0.72 HTT (0.59) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL4342223 0.72 HTT (0.59) HTTPOLBMAPTALDH1A1MEN1
SCHEMBL9355395 0.70 HTT (0.47) HTTPOLBMAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed