SCHEMBL4358931

SCHEMBL4358931

O=C(Nc1ccc(C(F)(F)F)cc1)N(S)c1cc(F)c(O)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
MTOR P42345 4/20 0.45
BAZ1A Q9NRL2 1/20 0.45
KIF11 P52732 1/20 0.43
TGM2 P21980 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 1/20 0.43
P2RX1 P51575 1/20 0.42
P2RX4 Q99571 1/20 0.42
P2RX7 Q99572 1/20 0.42
TMPRSS4 Q9NRS4 1/20 0.42
TRPV1 Q8NER1 2/20 0.41
PTGS1 P23219 2/20 0.41
RORC P51449 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4342201 0.88 EPHX2 (0.45) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4353865 0.86 EPHX2 (0.46) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4359460 0.86 EPHX2 (0.46) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4346166 0.83 TSHR (0.49) EPHX2NPC1RAB9AALDH1A1P2RX1
SCHEMBL4341297 0.82 KMT2A (0.43) EPHX2MTORNPC1RAB9AALDH1A1
SCHEMBL4348981 0.81 EPHX2 (0.43) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4347077 0.80 EPHX2 (0.45) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4348054 0.80 EPHX2 (0.45) EPHX2MTORBAZ1AKIF11TGM2
SCHEMBL4341863 0.80 HDAC3 (0.48) EPHX2MTORTRPV1
SCHEMBL4341321 0.79 P2RX1 (0.50) EPHX2MTORBAZ1AKIF11TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed