SCHEMBL4362902

SCHEMBL4362902

COC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.71
HRH4 Q9H3N8 5/20 0.67
HRH3 Q9Y5N1 2/20 0.65
POLB P06746 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
RBP4 P02753 1/20 0.60
DRD3 P35462 2/20 0.56
ADRB1 P08588 1/20 0.56
HTR1A P08908 1/20 0.56
ADRA2C P18825 1/20 0.56
HTR2B P41595 1/20 0.56
TMEM97 Q5BJF2 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
PDE4B Q07343 1/20 0.56
GRIN2D O15399 1/20 0.56
GRIN3B O60391 1/20 0.56
GRIN1 Q05586 1/20 0.56
GRIN2A Q12879 1/20 0.56
GRIN2B Q13224 1/20 0.56
GRIN2C Q14957 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11981458 0.83 AKR1C3 (1.00) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL23493748 0.83 AKR1C3 (0.52) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL12803717 0.83 AKR1C3 (0.67) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL2350768 0.82 HRH4 (0.78) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL4368875 0.82 AKR1C3 (0.70) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL27306947 0.82 AKR1C3 (0.66) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL31487392 0.82 AKR1C3 (0.70) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL12964356 0.82 AKR1C3 (0.68) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL15962961 0.81 AKR1C3 (0.80) AKR1C3HRH4HRH3POLBSMN1; SMN2
SCHEMBL1810411 0.81 DRD3 (0.64) AKR1C3HRH4HRH3POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010487-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. Hoffmann-Roche AG (CH) 2009-01-07 EP disclosed
WO-2007115938-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO disclosed