SCHEMBL436580

SCHEMBL436580

O=C(OCc1ccc(-c2noc(CCC3(c4cccc(C(F)(F)F)c4)CCOCC3)n2)cc1)C1CNC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.49
HDAC1 Q13547 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
FFAR1 O14842 3/20 0.41
MAPT P10636 3/20 0.39
TSHR P16473 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
S1PR3 Q99500 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459650 0.81 S1PR1 (0.59) S1PR1MAPTTSHRHTTSMN1; SMN2
SCHEMBL436579 0.81 S1PR1 (0.73) S1PR1S1PR3
SCHEMBL16649407 0.79 S1PR1 (0.60) S1PR1HDAC1HDAC8HDAC6FFAR1
SCHEMBL435271 0.74 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL16649359 0.71 S1PR1 (0.54) S1PR1HDAC1HDAC8HDAC6FFAR1
SCHEMBL877139 0.67 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL436892 0.65 EPHX2 (0.52) FFAR1
SCHEMBL876952 0.65 S1PR1 (0.82) S1PR1S1PR3
SCHEMBL461254 0.65 S1PR1 (0.86) S1PR1S1PR3
SCHEMBL459685 0.65 S1PR1 (0.72) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595969-A1 SUBSTITUTED 3-PHENYL-1,2,4-OXADIAZOLE COMPOUNDS Bristol-Myers Squibb Company (US) 2013-05-29 EP disclosed
WO-2012012477-A1 SUBSTITUTED 3-PHENYL-1,2,4-OXADIAZOLE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-01-26 WO disclosed