SCHEMBL4369322

SCHEMBL4369322

COc1ccc2nccc(N3CCC(CNC4CCN(c5ccnc6ccc(OC)nc56)C4)C3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP8B1 Q9UNU6 1/20 0.43
KCNH2 Q12809 8/20 0.42
SLC2A1 P11166 1/20 0.40
ACVR1 Q04771 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13527138 0.86 KCNH2 (0.44) CYP8B1KCNH2SLC2A1
SCHEMBL1224389 0.85 CYP8B1 (0.47) CYP8B1KCNH2
SCHEMBL1224386 0.85 CYP8B1 (0.47) CYP8B1KCNH2
SCHEMBL14441508 0.84 CYP8B1 (0.44) CYP8B1KCNH2SLC2A1
SCHEMBL3665601 0.84 CYP8B1 (0.46) CYP8B1KCNH2ACVR1
SCHEMBL1224385 0.84 CYP8B1 (0.46) CYP8B1KCNH2ACVR1
SCHEMBL3179377 0.84 CYP8B1 (0.46) CYP8B1KCNH2ACVR1
SCHEMBL3259301 0.81 MAP4K4 (0.44) CYP8B1KCNH2SLC2A1
SCHEMBL1222880 0.80 CYP8B1 (0.48) CYP8B1
SCHEMBL4070886 0.80 CYP8B1 (0.45) CYP8B1KCNH2ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773343-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2009-05-13 EP disclosed
EP-1773343-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-04-18 EP disclosed
WO-2006017326-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2006-02-16 WO disclosed