SCHEMBL4370532

SCHEMBL4370532

CC1(C)CC(=O)c2c(C(F)(F)F)nn(-c3ccc(C#N)c(NC4CCNCC4)c3)c2C1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 19/20 0.60
HSP90AA1 P07900 17/20 0.60
HSP90B1 P14625 1/20 0.60
TRAP1 Q12931 1/20 0.60
OPRM1 P35372 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27196733 0.91 HSP90AB1 (0.61) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL13740696 0.90 HSP90AB1 (0.65) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL30839279 0.90 HSP90AB1 (0.74) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3631667 0.90 HSP90AB1 (0.65) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL1220779 0.90 HSP90AB1 (0.60) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL3633252 0.87 HSP90AB1 (0.59) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL1747106 0.85 HSP90AA1 (0.84) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL4380174 0.84 HSP90AB1 (0.58) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL13740369 0.84 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL13740368 0.84 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009114470-A2 TETRAHYDROINDOLE AND TETRAHDYROINDAZOLE AS HSP90 INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-09-17 WO disclosed