SCHEMBL4370923

SCHEMBL4370923

CCS(=O)(=O)N=C1NC(=O)C(=Cc2ccc3c(c2)OCO3)S1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.67
CSNK2A2 P19784 6/20 0.64
CSNK2B P67870 6/20 0.64
CSNK2A1 P68400 6/20 0.64
DYRK1A Q13627 6/20 0.64
CSNK2A3 Q8NEV1 6/20 0.64
DYRK1B Q9Y463 6/20 0.64
MAPK9 P45984 1/20 0.60
GSK3B P49841 1/20 0.54
PIM1 P11309 6/20 0.53
DYRK2 Q92630 6/20 0.53
DYRK3 O43781 5/20 0.53
CDK5 Q00535 3/20 0.53
CDK5R1 Q15078 3/20 0.53
KDM4E B2RXH2 3/20 0.51
MAPT P10636 3/20 0.51
HPGD P15428 3/20 0.51
KMT2A Q03164 3/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10093411 1.00 CDC25B (0.67) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL496829 0.88 DYRK1A (0.67) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL496943 0.88 DYRK1A (0.67) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL10093420 0.84 CDC25B (0.81) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL4379157 0.84 CDC25B (0.81) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL497117 0.84 CDC25B (0.81) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL497258 0.83 KMT2A (0.66) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL497260 0.83 KMT2A (0.66) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL497128 0.82 DYRK1A (0.71) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A
SCHEMBL496852 0.82 DYRK1A (0.71) CDC25BCSNK2A2CSNK2BCSNK2A1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648452-B1 2-IMINO-4-(THIO)OXO-5-POLYCYCLOVINYLAZOLINES FOR USE AS PI3 KINASE INHIBITORS MERCK SERONO SA (CH) 2009-07-22 EP claimed