SCHEMBL4375983

SCHEMBL4375983

O=c1c(NCc2ccccc2)c(Nc2ccncc2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 7/20 1.00
AURKB Q96GD4 10/20 0.74
ROCK1 Q13464 9/20 0.74
GSK3A P49840 8/20 0.74
GSK3B P49841 8/20 0.74
CDC42BPA Q5VT25 8/20 0.74
CSNK1G3 Q9Y6M4 8/20 0.74
CHEK2 O96017 7/20 0.74
PRKACA P17612 7/20 0.74
RPS6KB1 P23443 7/20 0.74
RPS6KA3 P51812 7/20 0.74
PRKG1 Q13976 6/20 0.74
PKN2 Q16513 6/20 0.74
HIPK4 Q8NE63 6/20 0.74
CSNK1G1 Q9HCP0 6/20 0.74
CHEK1 O14757 5/20 0.74
MKNK2 Q9HBH9 5/20 0.74
SGK2 Q9HBY8 5/20 0.74
AKT1 P31749 5/20 0.74
CSNK1G2 P78368 5/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4376451 0.92 MAPKAPK2 (0.85) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4030799 0.88 FLT4 (0.78) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4368914 0.85 ROCK1 (0.74) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4370778 0.85 GSK3A (1.00) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4369926 0.85 ROCK1 (0.74) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4374703 0.85 ROCK1 (1.00) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4364173 0.85 FLT4 (0.79) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4366308 0.83 ROCK1 (0.71) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4540504 0.82 GSK3A (0.75) MAPKAPK2AURKBROCK1GSK3AGSK3B
SCHEMBL4378368 0.81 ROCK1 (0.73) MAPKAPK2AURKBROCK1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO claimed
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed