SCHEMBL4378796

SCHEMBL4378796

Cc1ccc(CNC(C)C)cc1-n1c(C)cc(OCc2ccc(F)cc2F)c(Br)c1=O

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 20/20 0.66
ROCK2 O75116 1/20 0.66
MAPK12 P53778 1/20 0.66
MAPK11 Q15759 1/20 0.66
STRADA Q7RTN6 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL29593781 0.99 MAPK14 (0.65) MAPK14ROCK2MAPK12MAPK11STRADA
Hydrochloric Acid SCHEMBL4381791 0.99 MAPK14 (0.65) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4377211 0.86 MAPK14 (0.74) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL29594904 0.86 MAPK14 (0.74) MAPK14ROCK2MAPK12MAPK11STRADA
Hydrochloric Acid SCHEMBL6475356 0.85 MAPK14 (0.76) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL6499957 0.85 MAPK14 (0.80) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL5862122 0.85 MAPK14 (0.71) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4383268 0.85 MAPK14 (0.72) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL29594431 0.85 MAPK14 (0.71) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL5266295 0.84 MAPK14 (0.47) MAPK14ROCK2MAPK12MAPK11STRADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP claimed
CN-114748622-A P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD 弗尔康医疗公司 2022-07-15 CN disclosed
CN-114732910-A P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2022-07-12 CN disclosed
CN-111601593-B P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2022-04-15 CN disclosed
CN-111601593-A P38 kinase inhibitor reduces DUX4 and downstream gene expression for treatment of FSHD 弗尔康医疗公司 2020-08-28 CN disclosed
US-7629363-B2 antiinflammatory agent for treating asthma and chronic pulmonary inflammatory disease PFIZER INC (US) 2009-12-08 US disclosed
US-7629363-B2 antiinflammatory agent for treating asthma and chronic pulmonary inflammatory disease PFIZER INC (US) 2009-12-08 US disclosed
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP disclosed