SCHEMBL4379795

SCHEMBL4379795

CC(C)(NC(=O)n1c(=O)n(CC2CCCCC2)c2ccccc21)C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 11/20 0.51
CNR1 P21554 4/20 0.51
OPRL1 P41146 5/20 0.45
OPRM1 P35372 4/20 0.45
NPC1 O15118 1/20 0.43
OPRK1 P41145 1/20 0.43
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HTR3A P46098 1/20 0.41
HTR4 Q13639 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920069 0.97 CNR2 (0.52) CNR2CNR1OPRL1OPRM1TMEM97
SCHEMBL3918328 0.87 CNR2 (0.58) CNR2CNR1TMEM97SIGMAR1HTR3A
SCHEMBL14261065 0.84 CNR2 (0.48) CNR2CNR1OPRL1TMEM97SIGMAR1
SCHEMBL4382324 0.82 CNR2 (0.74) CNR2CNR1OPRL1OPRM1TMEM97
SCHEMBL14261351 0.79 CNR2 (0.65) CNR2CNR1OPRL1OPRM1TMEM97
SCHEMBL3916842 0.79 CNR2 (0.75) CNR2CNR1OPRL1TMEM97SIGMAR1
SCHEMBL3919334 0.79 CNR2 (0.62) CNR2CNR1OPRL1OPRM1TMEM97
SCHEMBL4392439 0.79 CNR2 (0.56) CNR2CNR1OPRL1OPRM1NPC1
SCHEMBL14261070 0.77 CNR2 (0.43) CNR2CNR1OPRL1OPRM1NPC1
SCHEMBL4385562 0.77 CNR2 (0.52) CNR2CNR1OPRL1OPRM1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090298811-A1 BENZIMIDAZOLONE DERIVATIVES PFIZER INC 2009-12-03 US claimed
US-20090298811-A1 BENZIMIDAZOLONE DERIVATIVES PFIZER INC 2009-12-03 US disclosed
WO-2008032164-A2 BENZIMIDAZOLONE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-03-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090298811-A1 BENZIMIDAZOLONE DERIVATIVES TRPV1, CNR1, CNR2 CNR2 3/4885CNR1 2/4885OPRL1 52/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.