SCHEMBL4381257

SCHEMBL4381257

CN(CCN(C)c1ccc(F)cc1F)CCn1ccc2c(-c3ccoc3C(=O)NN)nc(N)nc21

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 1/20 0.34
HDAC6 Q9UBN7 2/20 0.33
HDAC4 P56524 1/20 0.33
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850900 0.78 HDAC1 (0.44) HDAC1HDAC2HDAC6HDAC4
SCHEMBL2849515 0.78 ADA (0.41) HDAC1HDAC2ADORA2AADORA1
SCHEMBL4381259 0.76 MAPT (0.37) HDAC1HDAC2ADORA2AADORA1
SCHEMBL2843175 0.69 ADORA2A (0.49) HDAC1ADORA2AADORA1
SCHEMBL28806935 0.61 ADORA2A (0.43) HDAC1ADORA2A
SCHEMBL14019391 0.60 ADORA2A (0.50) HDAC1ADORA2AADORA1
SCHEMBL27932477 0.59 PIK3CA (0.34) ADORA2APIK3CA
SCHEMBL27932436 0.59 ADORA2A (0.34) HDAC1ADORA2APIK3CAMTOR
SCHEMBL27914295 0.59 ADORA2A (0.35) HDAC1ADORA2A
SCHEMBL14922346 0.58 ADORA2A (0.62) HDAC1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2129220-A2 ADENOSINE A2A RECEPTOR ANTAGONISTS King Pharmaceuticals Research and Development Inc. (US) 2009-12-09 EP disclosed
WO-2008121748-A2 ADENOSINE A2A RECEPTOR ANTAGONISTS KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT,INC. (US) 2008-10-09 WO disclosed