SCHEMBL4387428

SCHEMBL4387428

COC(=O)c1ccc(Cn2nc(-c3cc(F)c(F)c(F)c3)cc2C(=O)NC2CCC(C(C)(C)C)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.46
BRD4 O60885 1/20 0.43
GIPR P48546 1/20 0.43
CNR2 P34972 6/20 0.42
CNR1 P21554 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
SMYD3 Q9H7B4 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884636 1.00 GCGR (0.47) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL2883065 0.92 PTGDR2 (0.49) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL2885559 0.92 PTGDR2 (0.49) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL13632823 0.92 PTGDR2 (0.47) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL2883069 0.92 PTGDR2 (0.49) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL2882637 0.87 GCGR (0.58) GCGRPTGDR2GIPR
SCHEMBL2666811 0.87 GCGR (0.58) GCGRPTGDR2GIPR
SCHEMBL2666818 0.87 GCGR (0.58) GCGRPTGDR2GIPR
SCHEMBL2878249 0.84 GCGR (0.45) GCGRPTGDR2BRD4GIPRCNR2
SCHEMBL2666584 0.84 GCGR (0.45) GCGRPTGDR2BRD4GIPRCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765335-B1 PYRAZOLE AMIDE DERIVATIVES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO INC (US) 2009-11-25 EP disclosed