SCHEMBL4399892

SCHEMBL4399892

O=C(O)N(CCCN(Cc1ccc(-n2cncn2)cc1)C(=O)OCc1cncs1)Cc1ccc(-n2cncn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.44
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
PTGER2 P43116 1/20 0.34
NPC1 O15118 2/20 0.34
LMNA P02545 1/20 0.34
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL893312 0.97 CYP3A4 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19POLB
SCHEMBL892850 0.90 CYP3A4 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19POLB
SCHEMBL894408 0.87 CYP3A4 (0.38) CYP3A4CYP2D6CYP2C9CYP2C19POLB
SCHEMBL9943431 0.85 CYP3A4 (0.40) CYP3A4CYP2D6CYP2C9CYP2C19POLB
SCHEMBL4248044 0.83 CYP3A4 (0.57) CYP3A4CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9943460 0.82 CYP3A4 (0.39) CYP3A4CYP2D6CYP2C9CYP2C19POLB
SCHEMBL4398374 0.81 CYP3A4 (0.52) CYP3A4CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL893063 0.81 CYP3A4 (0.59) CYP3A4CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL4252360 0.81 CYP3A4 (0.49) CYP3A4CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL4390638 0.80 CYP3A4 (0.51) CYP3A4CYP2D6CYP2C9CYP2C19TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed
EP-2465855-A1 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed