SCHEMBL4405909

SCHEMBL4405909

COc1ccc(C(C)C)cc1-c1cc2c(cn1)[nH]c(=O)n2C1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.45
CHRM2 P08172 3/20 0.43
CHRM4 P08173 3/20 0.43
CHRM1 P11229 3/20 0.43
CHRM5 P08912 2/20 0.43
CHRM3 P20309 2/20 0.43
KCNH2 Q12809 2/20 0.43
JAK2 O60674 7/20 0.41
JAK3 P52333 7/20 0.41
JAK1 P23458 1/20 0.41
OPRM1 P35372 4/20 0.38
MAP3K11 Q16584 1/20 0.38
PRKDC P78527 1/20 0.37
ATM Q13315 1/20 0.37
ATR Q13535 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481589 0.81 MTOR (0.55) BRD4JAK2JAK3JAK1MAP3K11
SCHEMBL481329 0.76 MAP3K11 (0.50) MAP3K11
SCHEMBL481330 0.76 MAP3K11 (0.50) MAP3K11
SCHEMBL481687 0.76 MAP3K11 (0.50) MAP3K11
SCHEMBL4635792 0.72 CHRM1 (0.74) CHRM2CHRM4CHRM1CHRM5CHRM3
SCHEMBL481598 0.72 MAP3K11 (0.62) MAP3K11
Hydrochloric Acid SCHEMBL4635941 0.72 CHRM1 (0.72) CHRM2CHRM4CHRM1CHRM5CHRM3
SCHEMBL481696 0.72 MAP3K11 (0.61) JAK2JAK3JAK1MAP3K11
SCHEMBL481851 0.71 MAP3K11 (0.53) JAK2JAK3JAK1MAP3K11
SCHEMBL15205927 0.71 FYN (0.38) BRD4MAP3K11PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2090577-A2 Heteroaryl compounds, compositions thereof, and their use as protein kinase inhibitors Signal Pharmaceuticals LLC (US) 2009-08-19 EP claimed