SCHEMBL4410643

SCHEMBL4410643

[CH2]Cn1c(=O)c(C(C)=O)c(NC(C)=O)c2cc(-c3ccc(Cl)cc3)c(-c3ccc(Cl)cc3Cl)nc21

nearest known ligand 0.84

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.84
CNR2 P34972 19/20 0.84
GABRA1 P14867 2/20 0.79
ADRA2C P18825 2/20 0.79
SLC6A3 Q01959 2/20 0.79
EGFR P00533 1/20 0.79
ALOX5 P09917 1/20 0.79
ADORA3 P0DMS8 1/20 0.79
MAPK3 P27361 1/20 0.79
OPRL1 P41146 1/20 0.79
SLC18A2 Q05940 1/20 0.79
MAPK14 Q16539 1/20 0.79
TMEM97 Q5BJF2 1/20 0.79
SIGMAR1 Q99720 1/20 0.79
ADRB3 P13945 1/20 0.62
ADRA2B P18089 1/20 0.62
HTR2A P28223 1/20 0.62
HTR2C P28335 1/20 0.62
OPRD1 P41143 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3622197 0.93 CNR1 (0.87) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3624716 0.91 CNR1 (1.00) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3625806 0.90 CNR1 (0.89) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3627977 0.90 CNR1 (1.00) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3616947 0.89 CNR1 (0.86) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3624317 0.89 CNR1 (1.00) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3621869 0.88 CNR1 (0.80) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL4396445 0.88 CNR1 (0.86) CNR1CNR2GABRA1ADRA2CSLC6A3
SCHEMBL3621918 0.88 CNR1 (1.00) CNR1CNR2GABRA1ADRA2CSLC6A3
Naphthyridinone SCHEMBL762298 0.88 CNR1 (1.00) CNR1CNR2GABRA1ADRA2CSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682550-B1 SUBSTITUTED NAPHTHYRIDINONE DERIVATIVES MERCK & CO INC (US) 2009-12-23 EP claimed