SCHEMBL4419970

SCHEMBL4419970

CCN=CN(C)c1cc(C)c(Oc2ccc(F)c(C(F)(F)F)c2)cc1C

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
SLC6A4 P31645 2/20 0.40
KCNH2 Q12809 1/20 0.40
AR P10275 14/20 0.34
RHEB Q15382 1/20 0.32
BRAF P15056 1/20 0.32
KDR P35968 1/20 0.32
SCN9A Q15858 1/20 0.31
PLA2G7 Q13093 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427117 0.88 SCN9A (0.38) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL4414450 0.86 AR (0.53) AR
SCHEMBL6905031 0.81 GRIN2B (0.31)
SCHEMBL17222147 0.81 HTR2A (0.40) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL6907658 0.78 MRGPRX4 (0.33)
SCHEMBL4428667 0.77 HTR2A (0.40) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL119682 0.77 HTR2A (0.40) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL29427853 0.77 HTR2A (0.40) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL1278451 0.77 HTR2A (0.40) HTR2ASLC6A4KCNH2ARRHEB
SCHEMBL28347300 0.75 HTR2A (0.41) HTR2ASLC6A4KCNH2ARRHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562569-B1 ANTIFUNGAL MEDICAMENTS COMPRISING ARYLAMIDINE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2009-12-23 EP claimed