SCHEMBL4420175

SCHEMBL4420175

COc1ccc(-c2nc(-c3ccc4c(c3)CCN4)no2)cc1C#N

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.64
S1PR3 Q99500 7/20 0.64
KCNH2 Q12809 3/20 0.49
NPC1 O15118 1/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4426038 0.89 S1PR1 (0.78) S1PR1S1PR3KCNH2
SCHEMBL2982991 0.87 S1PR1 (0.80) S1PR1S1PR3KCNH2
Hydrochloric Acid SCHEMBL2991865 0.86 S1PR1 (0.79) S1PR1S1PR3KCNH2
SCHEMBL566253 0.84 S1PR1 (0.67) S1PR1S1PR3NPC1MAPTSMN1; SMN2
SCHEMBL566042 0.78 S1PR1 (1.00) S1PR1S1PR3NPC1MAPTSMN1; SMN2
SCHEMBL566600 0.78 S1PR1 (0.59) S1PR1S1PR3NPC1MAPTSMN1; SMN2
SCHEMBL2602064 0.76 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL2121369 0.76 S1PR1 (0.76) S1PR1S1PR3KCNH2SMN1; SMN2
SCHEMBL566029 0.76 S1PR1 (0.59) S1PR1S1PR3NPC1MAPTSMN1; SMN2
SCHEMBL566290 0.76 S1PR1 (0.76) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151621-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed