SCHEMBL4420561

SCHEMBL4420561

CNC(=O)CNc1cc(-c2ccsc2)ccc1N

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.52
KCNH2 Q12809 2/20 0.48
HDAC2 Q92769 4/20 0.46
CHEK2 O96017 2/20 0.42
HDAC3 O15379 3/20 0.39
ACMSD Q8TDX5 1/20 0.39
CYP1A2 P05177 1/20 0.38
GSK3B P49841 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
TRPM4 Q8TD43 1/20 0.38
IKBKB O14920 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653316 0.85 HDAC1 (0.70) HDAC1KCNH2HDAC2HDAC3HDAC6
SCHEMBL4579995 0.77 HDAC1 (0.75) HDAC1KCNH2HDAC2HDAC3MAPT
SCHEMBL4312605 0.72 HDAC1 (0.53) HDAC1KCNH2HDAC2CHEK2HDAC3
SCHEMBL650082 0.72 HDAC1 (0.74) HDAC1KCNH2HDAC2HDAC3HDAC6
SCHEMBL3643629 0.71 HDAC1 (0.77) HDAC1KCNH2HDAC2HDAC3HDAC6
SCHEMBL3643627 0.71 HDAC1 (0.73) HDAC1KCNH2HDAC2HDAC3
SCHEMBL4120548 0.70 HDAC1 (0.76) HDAC1KCNH2HDAC2HDAC3
SCHEMBL9983570 0.70 HDAC1 (0.49) HDAC1HDAC2HDAC3ALDH1A1HDAC6
SCHEMBL4578938 0.69 HDAC1 (0.74) HDAC1KCNH2HDAC2HDAC3
SCHEMBL3774949 0.69 HDAC1 (0.74) HDAC1KCNH2HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013196-A2 DISUBSTITUTED ANILINE COMPOUNDS Merck & Co., Inc. (US) 2009-01-14 EP disclosed
WO-2007127137-A2 DISUBSTITUTED ANILINE COMPOUNDS MERCK & CO., INC. (US) 2007-11-08 WO disclosed