SCHEMBL4422579

SCHEMBL4422579

O=C(O)N1CCC2(CCn3c(nc(-c4ccncc4)cc3=O)N2C[C@H](O)c2ccccc2)C1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.45
USP19 O94966 4/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
CYP1A2 P05177 4/20 0.36
CYP2D6 P10635 4/20 0.36
CYP2C9 P11712 4/20 0.36
USP2 O75604 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4422570 1.00 GSK3B (0.45) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL5554351 0.94 GSK3B (0.46) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL5554356 0.94 GSK3B (0.46) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL4421910 0.91 GSK3B (0.42) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL4421905 0.91 GSK3B (0.42) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL4416870 0.90 KDM4E (0.43) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL4416876 0.90 KDM4E (0.43) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL3365321 0.90 GSK3B (0.50) GSK3BPIK3R1PIK3CACYP1A2CYP2D6
SCHEMBL4430878 0.89 GSK3B (0.41) GSK3BUSP19ALDH1A1TSHRPIK3R1
SCHEMBL4430874 0.89 GSK3B (0.41) GSK3BUSP19ALDH1A1TSHRPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547705-B2 Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives SANOFI-AVENTIS (FR) 2009-06-16 US claimed
EP-1557417-B1 Substituted 8'-pyri(mi)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a] pyrimidin-6-one derivatives SANOFI AVENTIS (FR) 2007-03-07 EP claimed