SCHEMBL4423344

SCHEMBL4423344

O=c1ccc(C(c2ccccc2)c2ccccc2)nn1CC1CCCCC1Cc1cccc(O)c1.[NaH]

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.43
PTGDR2 Q9Y5Y4 2/20 0.42
PTGDR Q13258 1/20 0.41
CYP19A1 P11511 1/20 0.40
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
OPRM1 P35372 6/20 0.34
OPRD1 P41143 6/20 0.34
OPRK1 P41145 6/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
MMP2 P08253 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3159504 0.83 PTGDR2 (0.65) PTGIRPTGDR2PTGDR
SCHEMBL16493870 0.68 PTGDR2 (0.48) PTGIRPTGDR2PTGDRCYP19A1ALDH1A1
SCHEMBL3169598 0.67 ESR1 (0.48) CYP19A1OPRM1OPRD1OPRK1
SCHEMBL3176694 0.66 PTGDR2 (0.51) PTGIRPTGDR2PTGDRCYP19A1ALDH1A1
SCHEMBL7772431 0.66 PTGIR (0.73) PTGIRPTGDRCYP19A1
SCHEMBL12198738 0.64 PTGIR (0.60) PTGIRPTGDR2PTGDR
SCHEMBL2510624 0.64 PTGIR (0.60) PTGIRPTGDR2PTGDR
SCHEMBL7777390 0.63 PTGIR (0.47) PTGIRPTGDR2PTGDR
SCHEMBL3178973 0.63 PTGDR2 (0.76) PTGIRPTGDR2PTGDRSMN1; SMN2PDE4A
SCHEMBL3174326 0.62 PTGDR2 (0.56) PTGIRPTGDR2PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094662-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS Astellas Pharma Inc. (JP) 2009-09-02 EP disclosed
WO-2008072784-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS ASTELLAS PHARMA INC. (JP) 2008-06-19 WO disclosed