SCHEMBL4425855

SCHEMBL4425855

O=C(O)N1CCC2(CCn3c(nc(-c4ccncn4)cc3=O)N2C[C@H](O)c2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.43
CYP2D6 P10635 4/20 0.40
CYP1A2 P05177 1/20 0.37
CYP46A1 Q9Y6A2 1/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4425837 1.00 GSK3B (0.43) GSK3BCYP2D6CYP1A2CYP46A1PIK3R1
SCHEMBL4425851 1.00 GSK3B (0.43) GSK3BCYP2D6CYP1A2CYP46A1PIK3R1
SCHEMBL5559223 0.95 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP46A1
SCHEMBL5559206 0.95 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP46A1
SCHEMBL5559215 0.95 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP46A1
SCHEMBL4421017 0.91 GSK3B (0.42) GSK3BCYP2D6CYP1A2PIK3R1PIK3CA
SCHEMBL4421015 0.91 GSK3B (0.42) GSK3BCYP2D6CYP1A2PIK3R1PIK3CA
SCHEMBL5559918 0.90 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL4431960 0.90 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL5560982 0.90 GSK3B (0.42) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547705-B2 Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives SANOFI-AVENTIS (FR) 2009-06-16 US claimed
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP claimed