SCHEMBL4426486

SCHEMBL4426486

Cc1ccc(C(=O)Nc2cc(-c3ccsc3)ccc2N)cn1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.71
HDAC2 Q92769 9/20 0.57
KCNH2 Q12809 2/20 0.57
HDAC3 O15379 7/20 0.51
CHEK2 O96017 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8229392 0.87 HDAC1 (0.68) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4426482 0.87 HDAC1 (0.68) HDAC1HDAC2KCNH2HDAC3
SCHEMBL3643629 0.85 HDAC1 (0.77) HDAC1HDAC2KCNH2HDAC3
SCHEMBL3643627 0.82 HDAC1 (0.73) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4120548 0.82 HDAC1 (0.76) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4316366 0.82 HDAC1 (0.62) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4419408 0.81 HDAC1 (0.73) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4578938 0.81 HDAC1 (0.74) HDAC1HDAC2KCNH2HDAC3
SCHEMBL2359218 0.80 HDAC1 (0.57) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4120547 0.80 HDAC1 (0.73) HDAC1HDAC2KCNH2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049124-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP disclosed
WO-2008010985-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2008-01-24 WO disclosed