SCHEMBL4427346

SCHEMBL4427346

CCn1cnc2c(=O)n(-c3ccc(Cl)cc3)c(CC3CCCC3)nc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.53
DRD5 P21918 5/20 0.53
GRM1 Q13255 1/20 0.38
YTHDC1 Q96MU7 1/20 0.38
PRKCA P17252 2/20 0.37
HIF1A Q16665 2/20 0.37
CNR1 P21554 2/20 0.37
CLK1 P49759 3/20 0.36
CLK2 P49760 3/20 0.36
CDK1 P06493 3/20 0.36
CCNB1 P14635 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
TSHR P16473 2/20 0.36
NPC1 O15118 1/20 0.36
CCNT1 O60563 1/20 0.36
EGFR P00533 1/20 0.36
CDK4 P11802 1/20 0.36
EIF2AK2 P19525 1/20 0.36
CCNA2 P20248 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4506947 0.99 DRD1 (0.55) DRD1DRD5GRM1YTHDC1PRKCA
SCHEMBL4521319 0.93 DRD1 (0.46) DRD1DRD5GRM1PRKCAHIF1A
SCHEMBL4519246 0.92 DRD1 (0.45) DRD1DRD5PRKCAHIF1ACNR1
SCHEMBL4559848 0.91 DRD1 (0.47) DRD1DRD5GRM1PRKCAHIF1A
SCHEMBL4521605 0.89 DRD1 (0.43) DRD1DRD5HIF1ACNR1CDK1
SCHEMBL4514450 0.85 DRD1 (0.38) DRD1DRD5GRM1PRKCAHIF1A
SCHEMBL4520124 0.83 DRD1 (0.53) DRD1DRD5GRM1CNR1CDK1
SCHEMBL4421685 0.83 DRD1 (0.51) DRD1DRD5GRM1PRKCAHIF1A
SCHEMBL5440724 0.83 PDE7A (0.46) DRD1DRD5GRM1YTHDC1PRKCA
SCHEMBL4413685 0.82 DRD1 (0.52) DRD1DRD5GRM1PRKCACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO claimed