SCHEMBL4428654

SCHEMBL4428654

COCCOc1ccc(-c2c(C#N)c(N)nc(SCc3csc(-c4cccs4)n3)c2C#N)cc1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 18/20 0.67
SLC6A3 Q01959 1/20 0.65
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
PKM P14618 1/20 0.54
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
MAPK10 P53779 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4426727 0.89 ADORA1 (0.82) ADORA1SLC6A3
SCHEMBL4432630 0.88 ADORA1 (0.71) ADORA1SLC6A3
SCHEMBL14464879 0.88 ADORA1 (0.84) ADORA1SLC6A3
SCHEMBL13929774 0.87 ADORA1 (0.65) ADORA1SLC6A3
SCHEMBL4427010 0.86 ADORA1 (0.74) ADORA1SLC6A3ALDH1A1KDM4EMEN1
SCHEMBL4428648 0.86 ADORA1 (0.85) ADORA1SLC6A3ALDH1A1SMN1; SMN2PKM
SCHEMBL4427399 0.86 ADORA1 (0.67) ADORA1SLC6A3ALDH1A1KDM4EMEN1
SCHEMBL4435702 0.86 ADORA1 (0.67) ADORA1SLC6A3ALDH1A1KDM4EMEN1
SCHEMBL13929511 0.84 ADORA1 (0.70) ADORA1SLC6A3ALDH1A1KDM4ELMNA
SCHEMBL13929983 0.84 ADORA1 (0.65) ADORA1SLC6A3ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455785-B1 SUBSTITUTED 2-THIO-3,5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THE USE OF THE SAME BAYER HEALTHCARE AG (DE) 2009-03-04 EP disclosed
EP-1455785-A1 SUBSTITUTED 2-THIO-3,5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THE USE OF THE SAME Bayer HealthCare AG (DE) 2004-09-15 EP disclosed
WO-2003053441-A1 SUBSTITUTED 2-THIO-3,5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THE USE OF THE SAME BAYER HEALTHCARE AG (DE) 2003-07-03 WO disclosed