SCHEMBL4429676

SCHEMBL4429676

O=C(CN(CC(=O)Nc1ccccc1)c1ccc(C(=O)Nc2ccccc2[AsH2])cc1)Nc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC3 O15379 2/20 0.48
NCOR2 Q9Y618 2/20 0.48
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
PTPN1 P18031 2/20 0.44
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
NOX1 Q9Y5S8 1/20 0.43
KCNK3 O14649 2/20 0.42
KCNK9 Q9NPC2 1/20 0.42
MDM4 O15151 1/20 0.42
TP53 P04637 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653999 0.85 HDAC1 (0.70) HDAC1HDAC2HDAC3NCOR2HDAC8
SCHEMBL651392 0.79 GAA (0.54) MEN1NPC1RAB9AKMT2ANOX1
SCHEMBL3836570 0.77 MEN1 (0.56) HDAC1MEN1NPC1RAB9AKMT2A
SCHEMBL651514 0.74 MEN1 (0.63) PTPN1MEN1NPC1RAB9AKMT2A
SCHEMBL8228268 0.73 HDAC1 (0.70) HDAC1HDAC2HDAC3HDAC8HDAC6
SCHEMBL3680858 0.73 KMT2A (0.71) HDAC2PTPN1HDAC8HDAC6MEN1
SCHEMBL13603928 0.73 KMT2A (0.57) MEN1NPC1RAB9AKMT2ANOX1
SCHEMBL889852 0.73 MEN1 (0.51) MEN1NPC1RAB9AKMT2ANOX1
SCHEMBL30451287 0.71 MEN1 (0.53) MEN1NPC1RAB9AKMT2ANOX1
SCHEMBL13644980 0.71 CA1 (0.50) MEN1NPC1RAB9AKMT2ANOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013196-A2 DISUBSTITUTED ANILINE COMPOUNDS Merck & Co., Inc. (US) 2009-01-14 EP disclosed
WO-2007127137-A2 DISUBSTITUTED ANILINE COMPOUNDS MERCK & CO., INC. (US) 2007-11-08 WO disclosed