SCHEMBL4430005

SCHEMBL4430005

CCC(CC)c1ccc(C(=O)Nc2cc(-c3ccccc3)ccc2N)cc1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.70
HDAC2 Q92769 10/20 0.70
HDAC3 O15379 3/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18653509 0.86 HDAC2 (0.75) HDAC1HDAC2HDAC3
SCHEMBL2209878 0.85 HDAC1 (0.62) HDAC1HDAC2HDAC3
SCHEMBL1689215 0.84 HDAC2 (0.75) HDAC1HDAC2HDAC3
SCHEMBL16380794 0.83 HDAC2 (1.00) HDAC1HDAC2HDAC3
SCHEMBL26775695 0.82 HDAC2 (0.86) HDAC1HDAC2HDAC3
SCHEMBL18653510 0.82 HDAC1 (0.73) HDAC1HDAC2HDAC3
SCHEMBL18653508 0.81 HDAC1 (0.76) HDAC1HDAC2HDAC3
SCHEMBL4581182 0.81 HDAC2 (0.83) HDAC1HDAC2HDAC3
SCHEMBL2209877 0.81 HDAC1 (0.59) HDAC1HDAC2HDAC3
SCHEMBL2108793 0.81 HDAC2 (0.65) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049124-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP disclosed
WO-2008010985-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2008-01-24 WO disclosed