SCHEMBL4430286

SCHEMBL4430286

CNC(=O)[C@H](NCC[C@H](c1ccc(C(F)(F)F)cc1)c1cccc(C)c1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
CCR2 P41597 9/20 0.45
ALDH1A1 P00352 2/20 0.43
CTDSP1 Q9GZU7 1/20 0.43
ALOX5 P09917 4/20 0.43
EPHX2 P34913 4/20 0.43
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
ALOX12 P18054 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
TACR1 P25103 1/20 0.41
TACR3 P29371 1/20 0.41
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4428071 1.00 KDM4E (0.48) KDM4ECCR2ALDH1A1CTDSP1ALOX5
Hydrochloric Acid SCHEMBL4431282 0.99 KDM4E (0.47) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4434552 0.91 CNR1 (0.51) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4427927 0.91 CNR1 (0.51) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4431735 0.91 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4433693 0.91 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4432388 0.90 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4430647 0.90 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4441795 0.90 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4432417 0.90 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed